Václav Bazgier
Václav Bazgier
E-mailová adresa ověřena na: upol.cz - Domovská stránka
NázevCitaceRok
A novel series of highly potent 2, 6, 9-trisubstituted purine cyclin-dependent kinase inhibitors
T Gucky, R Jorda, M Zatloukal, V Bazgier, K Berka, E Řezníčková, ...
Journal of medicinal chemistry 56 (15), 6234-6247, 2013
412013
Antiallergic effects of pigments isolated from green sea urchin (Strongylocentrotus droebachiensis) shells
ON Pozharitskaya, AN Shikov, MN Makarova, SA Ivanova, VM Kosman, ...
Planta medica 79 (18), 1698-1704, 2013
372013
Novel N-substituted indole Schiff bases as dual inhibitors of cyclooxygenase-2 and 5-lipoxygenase enzymes: Synthesis, biological activities in vitro and docking …
PF Lamie, WAM Ali, V Bazgier, L Rárová
European journal of medicinal chemistry 123, 803-813, 2016
312016
Synthesis, biological evaluation and molecular modeling of a novel series of 7-azaindole based tri-heterocyclic compounds as potent CDK2/Cyclin E inhibitors
CB Baltus, R Jorda, C Marot, K Berka, V Bazgier, V Kryštof, G Prié, ...
European journal of medicinal chemistry 108, 701-719, 2016
252016
MOLEonline: a web-based tool for analyzing channels, tunnels and pores (2018 update)
L Pravda, D Sehnal, D Toušek, V Navrátilová, V Bazgier, K Berka, ...
Nucleic acids research 46 (W1), W368-W373, 2018
212018
Synthesis and kinase inhibitory activity of new sulfonamide derivatives of pyrazolo [4, 3-e][1, 2, 4] triazines
M Mojzych, V Šubertová, A Bielawska, K Bielawski, V Bazgier, K Berka, ...
European journal of medicinal chemistry 78, 217-224, 2014
182014
Membrane-attached mammalian cytochromes P450: An overview of the membrane's effects on structure, drug binding, and interactions with redox partners
M Šrejber, V Navrátilová, M Paloncýová, V Bazgier, K Berka, ...
Journal of inorganic biochemistry 183, 117-136, 2018
122018
Acetylated deoxycholic (DCA) and cholic (CA) acids are potent ligands of pregnane X (PXR) receptor
A Carazo, L Hyrsova, J Dusek, H Chodounska, A Horvatova, K Berka, ...
Toxicology letters 265, 86-96, 2017
122017
Novel thidiazuron-derived inhibitors of cytokinin oxidase/dehydrogenase
J Nisler, D Kopečný, R Končitíková, M Zatloukal, V Bazgier, K Berka, ...
Plant molecular biology 92 (1-2), 235-248, 2016
112016
Biological activities of new monohydroxylated brassinosteroid analogues with a carboxylic group in the side chain
M Kvasnica, J Oklestkova, V Bazgier, L Rarova, K Berka, M Strnad
Steroids 85, 58-64, 2014
102014
2, 6, 9-Trisubstituted purines as CRK3 kinase inhibitors with antileishmanial activity in vitro
E Řezníčková, A Popa, T Gucký, M Zatloukal, L Havlíček, V Bazgier, ...
Bioorganic & medicinal chemistry letters 25 (11), 2298-2301, 2015
92015
Discovery of N2-(4-Amino-cyclohexyl)-9-cyclopentyl-N6-(4-morpholin-4-ylmethyl-phenyl)-9H-purine-2,6-diamine as a Potent FLT3 Kinase Inhibitor for Acute …
T Gucký, E Řezníčková, T Radošová Muchová, R Jorda, Z Klejová, ...
Journal of medicinal chemistry 61 (9), 3855-3869, 2018
82018
Characterization of a Pyrazolo[4,3‐d]pyrimidine Inhibitor of Cyclin‐Dependent Kinases 2 and 5 and Aurora A With Pro‐Apoptotic and Anti‐Angiogenic Activity In Vitro
E Řezníčková, S Weitensteiner, L Havlíček, R Jorda, T Gucký, K Berka, ...
Chemical biology & drug design 86 (6), 1528-1540, 2015
82015
Fluorone dyes have binding sites on both cytoplasmic and extracellular domains of Na, K-ATPase
M Havlíková, M Huličiak, V Bazgier, K Berka, M Kubala
Biochimica et Biophysica Acta (BBA)-Biomembranes 1828 (2), 568-576, 2013
72013
Exponential repulsion improves structural predictability of molecular docking
V Bazgier, K Berka, M Otyepka, P Banáš
Journal of computational chemistry 37 (28), 2485-2494, 2016
62016
Design, synthesis and biological activities of new brassinosteroid analogues with a phenyl group in the side chain
M Kvasnica, J Oklestkova, V Bazgier, L Rárová, P Korinkova, J Mikulík, ...
Organic & biomolecular chemistry 14 (37), 8691-8701, 2016
52016
Synthesis of novel aryl brassinosteroids through alkene cross-metathesis and preliminary biological study
P Korinkova, V Bazgier, J Oklestkova, L Rarova, M Strnad, M Kvasnica
Steroids 127, 46-55, 2017
42017
Arabidopsis histidine kinase 4 cytokinin receptor–the object of interest in ligand-receptor study
L Gallová, ZG Barreiro, V Bazgier, K Berka, P Mazura, L Spíchal, M Strnad
New Biotechnology, S165, 2016
22016
Channelsdb and moleonline-database and tool for analysis of biomacromolecular tunnels and pores
L Pravda, D Sehnal, K Berka, V Navrátilová, D Toušěk, V Bazgier, ...
Biophysical Journal 114 (3), 342a-343a, 2018
12018
Novel thiazolidinedione-hydroxamates as inhibitors of Mycobacterium tuberculosis virulence factor Zmp1
V Šlachtová, M Šebela, E Torfs, L Oorts, D Cappoen, K Berka, V Bazgier, ...
European journal of medicinal chemistry 185, 111812, 2020
2020
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Články 1–20